{"id":13,"date":"2016-03-06T17:59:05","date_gmt":"2016-03-06T16:59:05","guid":{"rendered":"https:\/\/filozofia.nett.to\/farmakologia\/2016\/03\/06\/analgetika-a-antiepileptika\/"},"modified":"2026-01-28T00:43:51","modified_gmt":"2026-01-27T23:43:51","slug":"analgetika-a-antiepileptika","status":"publish","type":"post","link":"https:\/\/filozofia.nett.to\/farmakologia\/sk\/analgetika-a-antiepileptika\/","title":{"rendered":"Analgetik\u00e1 a antiepileptik\u00e1"},"content":{"rendered":"<p><strong>Sodn\u00e1 so\u013e metamizolu:<\/strong> Okrem analg\u00e9zy m\u00e1 aj protiz\u00e1palov\u00e9 \u00fa\u010dinky. Presn\u00fd mechanizmus \u00fa\u010dinku nie je zn\u00e1my. Zatia\u013e sa hypoteticky predpoklad\u00e1, \u017ee metabolity tejto l\u00e1tky s\u00fa kanaboidy. Ak by to bola pravda, znamenalo by to, \u017ee t\u00e1to l\u00e1tka by mala nesmierne \u0161irok\u00e9 vyu\u017eitie<br \/>\nN02BB02 Sodn\u00e1 so\u013e metamizolu<br \/>\n<a href=\"https:\/\/en.wikipedia.org\/wiki\/Metamizole\" target=\"_blank\" rel=\"noopener\">https:\/\/en.wikipedia.org\/wiki\/Metamizole<\/a><br \/>\n*************************<br \/>\n<strong>Paracetamol<\/strong> tie\u017e moduluje endog\u00e9nnej kanabinoidn\u00fdch syst\u00e9m. Ovplyv\u0148uje iba CB1 receptor<br \/>\n*************************<br \/>\n<strong>flupirt\u00edn, Flupirtine<\/strong>, NMDA antagonista, GABAA modul\u00e1tor, obl\u00e1da dr\u00e1seln\u00fd kan\u00e1l<br \/>\n*************************<br \/>\n<strong>Pizotifen, pizotif\u00e9n<\/strong>, proti megr\u00e9nam, antagonista na dve typy seroton\u00ednov\u00fdch receptorov, antihistaminisk\u00e9 a anti-acetylchol\u00ednov\u00e9 \u00fa\u010dinky<br \/>\n*************************<br \/>\nN03AG04, <a href=\"https:\/\/en.wikipedia.org\/wiki\/Vigabatrin\" target=\"_blank\" rel=\"noopener\">https:\/\/en.wikipedia.org\/wiki\/Vigabatrin<\/a>, Vigabatrin, \u0161truktir\u00e1rne podobn\u00fd GABA<br \/>\n*************************<br \/>\n<a href=\"https:\/\/en.wikipedia.org\/wiki\/Gamma-Aminobutyric_acid\" target=\"_blank\" rel=\"noopener\">https:\/\/en.wikipedia.org\/wiki\/Gamma-Aminobutyric_acid<\/a>, Kyselina aminomaslov\u00e1 , ovplyv\u0148uje GABA svalov\u00fd tonus<br \/>\n*************************<br \/>\nFelbamate, Felbam\u00e1t, NMDA antagonista GABA agonista<br \/>\n*************************<br \/>\nLevetiracetam, \u0161truktur\u00e1rne podobn\u00fd Piracetamu, p\u00f4sob\u00ed na GABA a NMDA receptory<br \/>\n*************************<br \/>\nZonisamide, GABA, NMDA<br \/>\n*************************<br \/>\nPregabal\u00edn, <a href=\"https:\/\/en.wikipedia.org\/wiki\/Pregabalin\" target=\"_blank\" rel=\"noopener\">https:\/\/en.wikipedia.org\/wiki\/Pregabalin<\/a>, \u0161truktur\u00e1rne m\u00e1 ve\u013ea spolo\u010dn\u00e9ho s GABA<br \/>\n*************************<br \/>\n<a href=\"https:\/\/en.wikipedia.org\/wiki\/Perampanel\" target=\"_blank\" rel=\"noopener\">https:\/\/en.wikipedia.org\/wiki\/Perampanel<\/a>, Perampanel, selekt\u00edvny antagonista na AMPA receptory<br \/>\n*************************<br \/>\n<a href=\"https:\/\/en.wikipedia.org\/wiki\/Retigabine\" target=\"_blank\" rel=\"noopener\">https:\/\/en.wikipedia.org\/wiki\/Retigabine<\/a>, Retigabin, neeselekt\u00edvny NMDA<\/p>","protected":false},"excerpt":{"rendered":"Viacero druhov t\u00fdchto lie\u010div","protected":false},"author":1,"featured_media":0,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[2],"tags":[],"class_list":["post-13","post","type-post","status-publish","format-standard","hentry","category-farmakologia"],"_links":{"self":[{"href":"https:\/\/filozofia.nett.to\/farmakologia\/wp-json\/wp\/v2\/posts\/13","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/filozofia.nett.to\/farmakologia\/wp-json\/wp\/v2\/posts"}],"about":[{"href":"https:\/\/filozofia.nett.to\/farmakologia\/wp-json\/wp\/v2\/types\/post"}],"author":[{"embeddable":true,"href":"https:\/\/filozofia.nett.to\/farmakologia\/wp-json\/wp\/v2\/users\/1"}],"replies":[{"embeddable":true,"href":"https:\/\/filozofia.nett.to\/farmakologia\/wp-json\/wp\/v2\/comments?post=13"}],"version-history":[{"count":0,"href":"https:\/\/filozofia.nett.to\/farmakologia\/wp-json\/wp\/v2\/posts\/13\/revisions"}],"wp:attachment":[{"href":"https:\/\/filozofia.nett.to\/farmakologia\/wp-json\/wp\/v2\/media?parent=13"}],"wp:term":[{"taxonomy":"category","embeddable":true,"href":"https:\/\/filozofia.nett.to\/farmakologia\/wp-json\/wp\/v2\/categories?post=13"},{"taxonomy":"post_tag","embeddable":true,"href":"https:\/\/filozofia.nett.to\/farmakologia\/wp-json\/wp\/v2\/tags?post=13"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}